UtanoGadziriro

"Metadoksil": akaongororazve zvidhakwa, mirayiridzo kushandiswa, akafanana uye tsananguro

Sei zvinobudirira haazvibati zvinodhaka "Metadoksil"? Reviews yezvidhakwa, mari chigadzirwa ichi uye ayo zvinoratidza zvinokurukurwa pazasi. Uyewo munyaya ino, uchadzidza pamusoro nzira pokushandisa zvinodhaka, ayo nemishonga uye contraindications.

Description, chimiro, akafanana

Drug "Metadoksil" (zvidhakwa wongororo nezvazvo kucharatidzwa pazasi) rinowanikwa kutengeswa zvinotevera siyana:

  • Biconvex, rakatenderera chena mapiritsi pamwe Valium rumwe rutivi uye yakanyorwa zita chigadzirwa - panorumwe. Its vanoshingaira chirungiso ndiyo L maviri pyridoxine pyrrolidone carboxylate namashanu kana kunzi saka metadoksin. Uyewo vari vanobatanidzwa chokushandisa uyu MCC uye magnesium stearate.
  • The pachena mhinduro kuti jekiseni iri Hauoneki kana yellowish tint. chinoumba Its chikuru chiri metadoksin. Kunze pairi, muna zvinodhaka nziyo zvinosanganisira yavaibvisa edetate, D mvura / uye yavaibvisa metabisulfite uye methyl parahydroxybenzoate.

Chaizvoizvo zvinodhaka

"Metodoksil" - mushonga udhakwa. Ndizvo inzira yokuratidza detoxification uye hepatoprotective zvivako.

Hepatoprotective mugumisiro zvinodhaka nokuda kwayo Kamudzira tisazununguka. Uyezve, mushonga uyu anokwanisa kuderedza nhamba vakasununguka unsaturated uye zvine mafuta acids. Somugumisiro yakawedzera kuramba migumisiro hepatocyte peroxidation kwemafuta yomuka pasi pokudzora chepfu nevamiririri.

Detoxification ehupfumi zvinodhaka nokuda activation kuti chiropa makemikari izvo zvinobatanidzwa muviri panyaya iyi (zvikurukuru doro dehydrogenase uye acetaldehyde dehydrogenase), yekudyidzana Inowedzera muitiro yawo nokubviswa kubva mumuviri uye, sezvo zvakaguma izvozvo kunoderedza muchetura mugumisiro.

Features zvinodhaka

Chii chinoshamisa zvinodhaka "Metadoksil"? Instruction ratings vanoti chacho vanoshingaira fuma kunodzivisa paumbwe zvinhu zvakadai collagen uye fibronectin, uye chinonditadzisa kuunganidza triglycerides, izvo yekudyidzana DZEMUNHU DZINODZORA kukura cirrhosis.

Zvinofanira kucherechedzwa kuti chokushandisa ichi anokwanisa kupfupisa nguva zvakazorodza ucharwadziwa, kuderedza somatic uye mupfungwa zviratidzo hangover.

Hatigoni kutaura kuti metadoksin zvaanopa simba ari neGhebha-ergic uye cholinergic neurotransmitter hurongwa kunodzivisa gwenya excitation, anovandudza pfupi pakuyeuka uye mafungiro. Uyezve, imwe pfuma inokwanisa yokushandisa nayo ine nonspecific anxiolytic uye antidepressant zvinokonzerwa, uyewo kuderedza nehavi doro.

kinetics

Mushure kutora mushonga mukati riri kukurumidza woga kubva ura. Metadoksin ane refu bioavailability (vanenge 60-85%). Its ndichisunga kuti mapuroteni eplasma ndiyo 50%.

chikamu ichi rinoita ari chiropa yokuumba vanoshingaira nomukaka - pyrrolidone carboxylate uye pyridine.

Hafu-upenyu mushonga nokuda parenteral yaitonga kana ingestion maminitsi 45-57. Inenge 40-50% of zvinodhaka iri weti masikati uye vanenge 35-50% - ari mutsvina yadzo mumaawa 95.

umboo

Under chii ezvinhu inonyatsobudirira zvinodhaka achiita "Metadoksil"? Reviews zvidhakwa vanoti chingamubatsira uyu kwazvo chakanaka:

  • kudhakwa;
  • pakurapa chiropa chirwere, kusanganisira chidhakwa etiology;
  • doro kurega chirwere ;
  • doro kudhaka, kusanganisira chenjera.

Contraindications

mishonga tikaritora iri contraindicated mu:

  • achiyamwa;
  • gestation;
  • soro aikanganiswa pezvokuvamba zvinodhaka.

With inotarisirwa ichi rinofanira kushandiswa Parkinson, chirwere kunyanya kana murwere chava kushandisa levodopa. Izvi imhaka yokuti metadoksin anogona kuderedza kubudirira yokupedzisira.

Drug "Metadoksil": mirayiridzo kushandiswa

Reviews dzinoshuma kuti kushandiswa mari inofanira chete pashure zano nyanzvi.

Kana doro kudhaka, kunyanya chakasimba, kushingaira zvinodhaka chinotarisirwa intramuscularly panguva chipimo chemushonga ine 300-600 MG kana nomutsinga - 300-900 MG.

Kana achiita nomutsinga, zvinodhaka dose yakaratidza kare rakasanganiswa muna 5% dextrose mhinduro kana ne 500 ml yavaibvisa chloride. In chimiro kwakadaro kugadzirira kutaurwa dropwise, pamusoro maawa 1,4.

Sechikamu kurapa rechirume zvirwere chiropa, uye chisingaperi udhakwa ari mudziyo 500 MG raitongwa kaviri pazuva kwemaminitsi 25-35 pamberi kudya. dose Izvi zvinogona ngazviwedzerwe 500 MG katatu pazuva.

Nzira yokurapa pamwe zvinodhaka izvi zvinofanira kugara mazuva anenge 90.

Kana abstinent syndrome (doro) ari medicament chinotarisirwa nomutsinga nokuda aizomupa ari dose ine 900 MG kamwe pazuva kwemazuva 3-7 (zvichienderana murwere).

nemishonga

Chii kunaka vaite mushonga "Metadoksil"? Reviews yezvidhakwa rakashuma kuti akapoteredza kushandisa izvi zvinoreva kuti kazhinji kuva neutachiona.

Zvinofanira kucherechedzwa kuti vanhu bronchospasm kunogona kuitika chete Árbol asima (kakawanda kana uchishandisa mhinduro).

chaicho mashoko

Kuitwa "Metadoksil" jekiseni rine chinoumba akadai yavaibvisa metabisulfite. Izvi zvinhu zvinogona kukonzera asima kurwiswa mu muvamwe vanhu neutachiona, uyewo avo amplification.

Drug "Metadoksil": wongororo zvidhakwa

Zvinosuruvarisa wongororo kuti "Metadoksil" gadziriro, hapana zvikuru. Zvisinei, iwayo akasiya vanhu asingatani udhakwa, tinogona zvakachengeteka kugumisa kuti mushonga rinobatsira pakurapa doro nedoro.

Kana kubudirira kurapwa kuti ucharwadziwa, murwere inofambiswa ndiyo yakashatiswa mumufambiro chaizvo. Vamwe vanoti kana vagumirwe zvinodhaka kunobatsira kwazvo, apo vamwe - mukasazviziva zvainoita.

Uyewo rwawana kunaka mishumo mutengo chokushandisa ichi. Kazhinji, ndizvo 1250-1450 rubles.

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