UtanoGadziriro

The mushonga "Tizanil": mirayiridzo kushandiswa, analogs uye wongororo

"Tizanil" - mhasuru relaxant, ichipa musimboti chiito. Kuderedza mataurire skeletal tsandanyama kazhinji vakashandisa zvinodhaka "Tizanil" zvairatidza yokushandisa hunoita, kana zvakakodzera, kutsakatisa kwetsandanyama anovapo pave chetsinga chirwere chinopedza Disc chirwere, kuvhiya kana kukuvara. Kunze kushingaira chirungiso tizanidine, kuti medicament unotora mamwe zvinoriumba. Ebetsero nezvinozoitika nokuda pamberi nesilicon dioxide, stearic acid, microcrystalline cellulose uye lactose monohydrate.

Pharmacological chiito "Tizanila"

Alpha2-adrenergic receptors vari kusashanda paakaudzwa "Tizanil" zvinoreva. The Kuronga Pfungwa anogona kunyatsokurukura kubata acutely richiratidzwa chinyamunhari chinorwadza uye kurwadza kwacho mune chirwere chimiro, iye akavamba chepfungwa kana musana. mumiririri Izvi zvinobatsira kuderedza tsandanyama kuramba panguva pusa kufamba uye kuwedzera zvemasanga tsandanyama sunga.

Absorção de Água zvinodhaka kunoitika nokukurumidza. "Tizanil" mirayiridzo kushandiswa kwakafanana wezvinyorwa wefodya zvinenge zvachose kunonyanyisa mari yakawanikwa ropa maminitsi 60 tapinda zvomudumbu turakiti.

Muviri kunoitika muna chiropa, bioavailability anoenderana 34% tichisunga kuti yeplasma - 30%. Nokuti hafu-upenyu anotora avhareji yemaawa matatu. The mushonga iri yabudiswa kubva muviri sezvo metabolites kunyanya itsvo, mugove waro duku chinobviswa node.

umboo

Zvinoreva kuti "Tizanil" zvairatidza kuti kushandiswa ndeinotevera:

  • muzongoza chirwere pamwe kwetsandanyama, ayo achiperekedzwa nokurwadziwa;
  • chinorwadza kwetsandanyama pashure kuvhiyiwa;
  • skeletal tsandanyama spasticity somugumisiro chetsinga zvirwere.

Contraindications kugamuchira "Tizanila"

Mishonga contraindicated pamwe hypersensitivity kune yenhengo dzayo, kusagadzikana chiropa uye itsvo, wakati kududzwa. "Tizanil" kurayira haabvumiri kushandisa panguva gestation vomwana uye zamu achivadyisa. Contraindication ndiyo mishonga "fluvoxamine". Age isingasviki makore 18, kunorevawo kuti contraindications.

In renal insufficiency, mirayiridzo rinobvumira kushandiswa kwezvinodhaka, asi nokungwarira zvikuru. Izvi zvinoshandawo kwemajoini kushandiswa "Tizanila" ne CYP1A2 FIs uye kurapwa mune vakwegura.

Application medicament chipimo chemushonga

The mushonga chinobviswa nomuromo. Kana chinangwa kushandiswa kwezvinodhaka ndiko kubvisa kunorwadza kwetsandanyama, Zvinokurudzirwa kushandisa dose kubvira 2 kusvika 4 MG. Zvavakabvumirana dose ose nevamiririri zvinofanira kutorwa katatu pazuva. Kana nyaya rinorema, riri akabvumira kuwedzera imwe supplementation pamusoro 2-4 MG kuti medicament "Tizanil". Mahwendefa maererano application gwaro inogona kushandiswa skeletal tsandanyama spasticity 6mg. Ndicho vaifanira zuva chipimo chemushonga, izvo panguva kutanga kwekupwanyiwa kurapwa hakufaniri kupfuura. Mukurapa ezvinhu akadaro rinoitwa vatatu dosing nezuva. Kuchengeta penguva mazuva 3-7, iyo dose inogona zvishoma nezvishoma yakawedzera neavhareji 3 MG.

For kunonyanyisa zvazviri, vachiuya akabvumidza dose daily kusvika 24 MG. The optimum chipimo chemushonga iri kazhinji 12 MG kana kupfuura, asi haagoni pfuura 36 MG. Saka zuva nezuva zvinofanira kuitwa 3 kana 4 kugamuchirwa rinoreva "Tizanil". Mirayiridzo kushandiswa chine ruzivo pamusoro pakurapa varwere pamwe renal insufficiency. pakutanga varwere kwakadaro waitaura zvinodhaka kuti kushandiswa kamwe pazuva pane risingamboshandisi dose zvakafanana 2 MG. The chipimo chemushonga iri zvishoma nezvishoma zvakachinja maitiro murwere. Kana uchida kuwedzera dose, kuwedzera dose yokutanga, uye ipapo kushandura uwandu intakes.

nemishonga

kurapwa kwenguva refu dzimwe nguva aine zvisingadiwi zvinoitwa nhengo. Muchiitiko chino, vanogona kuva zvakawanda uye kuoneka kupfuura raidudzwa. Izvi zvinoshandawo negashiro guru mishonga kuti "Tizanil" chinodhaka. Mirayiridzo dzokushandisa Maererano izvi nemishonga, somunhu atadze kushanda zvakanaka pamusoro nemudumbu, vachiyanikira pamusoro mucous Kamudzira mumuromo, seasingakoshi kuderera BP, kurukutika, hope, dzungu nezvimwe nematambudziko zviitiko.

The kwaita nemishonga chikonzero kunorapwa kwachiremba, iyo kana kuderedza dose kana kubvisa chinodhaka, vachiitsiva nedzimwe nzira. In marapirwo mapiritsi "Tizanil" mirayiridzo kushandiswa kunge akacherechedza kuti ngozi nemishonga iri kushoma.

zvinodhaka kwavatori

The kukurukurirana mishonga yakasiyana - ichi chinokosha chaizvo mashoko, izvo zvinofanira kukurukurwa asati kurapwa kuderedza mukana wokuti nemishonga, kunze kukuvadza muviri uye yekuzvidzivirira kubudirira mishonga.

Zvinozivikanwa kuti zvinodhaka "Tizanil" pamwe "Fluvoxamine", unotungamirira Kuipa utano. Kana concomitantly chete antihypertensive zvinodhaka vanogona kuva bradycardia uye hypotension.

vose panyaya iyi kana sedatives uye mahwendefa kana "Tizanil" mirayiridzo kunoratidza kuwedzera nyaradzo, iyo anopiwa "Tizanilom". With pamwe yake mukanwa nhumbu anogona kutitadzisa Clearance hafu.

Drug kwavatori anogona kushandura efficacy kurapwa. With mawa kushandisa zvinodhaka akawanda, vanogona kuwedzera migumisiro mumwe kana inoodza mwoyo. Zvose izvi hwakazara chitarisiko nenjodzi, ovhadhozi, havana zvakakodzera mugumisiro.

Zvokungwarira

Asati atanga kurapwa ne "Tizanil" Zvinoratidza uye contraindications anofanira vainyatsoongorora.

It yakashuma panowanikwa rwakashata kuchinja itsvo chiropa. Asi mushonga kunobva achitora mushonga ari dose 12 MG zvichidzika, zviitiko zvakadaro zvakanga zvisingawanzoitiki.

Zvinonzi zano kuti nguva nenguva kutora chiropa shanda nemiedzo. Mumwedzi mina yokutanga - mwedzi kamwe. Mumamiriro ezvinhu umo AST uye alt mumatunhu mhiri kwomuzvarirwo tsika yekudyidzana kupfuudza navo, kunoda abolition zvinodhaka.

Vamwe varwere kutora "Tizanil" (kusanganisira analogs) anogona kuonekwa hope. Paaive mamiriro ichi, haugoni mabasa yaida wakawedzera kutarisirwa uye nokukurumidza siyana.

Nokuda mungozi Kushatiswa murwere zvinodhaka hauna akadzima pakarepo, zvinonzi kusiyiwa zvishoma nezvishoma dose rutapudzo.

Analogs "Tizanila"

Ushandiswe mune mirayiridzo yacho "Tizanil" kuverenga Hazviwanzovi kukubvumira kushandisa chepakuvamba nokuda zvimwe contraindications. Mishonga kupfuura anodhura ndezvaJehovha "tizanidine-din email" uye "Tizalud". mishonga ava zvakare relaxants, rinowanikwa piritsi muchimiro zvakafanana kushingaira chirungiso.

Kugadzirwa uye dzimwe analogs. Somuenzaniso, kunokwanisa "Mydocalm", "din email-Tizanilom" Surdaludom MR "," Surdaludom ".

Reviews

Reviews kuti "Tizanile" akasiyana, kureva. To. The mushonga kunogona kukanganisa varwere zvakasiyana. Asi kunyanya vari akanaka. Chivako ichi vakatanga kubudisa kwenguva refu, ndiko pasero kwenguva refu, vanhu vakawanda vakakwanisa nechokwadi kubudirira kwayo. Pane kunaka wongororo vasara nokuda nemigumisiro nokuda kusashivirirana yenhengo kana kushandiswa dzakakwirira mishonga pachii pakurapa "Tizanil" chinodhaka. Wongororo vakasara nevanhu vanofara pamwe mugumisiro, ari kurapwa kwacho zvinoenderana chipimo chemushonga chairayirwa chiremba, uye akapotsa haana kuona chero akaipa siyana.

mushonga aiwanzoshandisa kurapa chinopedza Disc chirwere. Pamusana chiito ayo zviratidzo pematanho chirwere kunyangarika nekukurumidza. Rasai nomusoro uye musana marwadzo, anovandudza kunopindirana utano. Dzimwe nguva pane kuduku divi Migumisiro akadai hope, kuoma kwezvinhu dzaiita zvokutaurwa mucosa, asi zvakakodzera kuchinja kubva dose kana kurega zvinodhaka zvingamera makumbo. Vamwe varwere chenjera ichiyerera osteochondrosis, kutsamwisa radicular urwere, kureva "Tizanil" vakadzokera chakaipa mufambo, apo vamwe mishonga haina kuuya unodikanwa zvabuda.

The mushonga hakuna kuipa anobvisa mukuru tsandanyama matauriro, razova migumisiro sitiroko. "Tizanil" vatora chete mushonga pamberi zvinoratidza zvakakodzera. Kana marapirwo kunodiwa munhu wechikuru kana murwere ane hosha chiropa, zviri nani kuti varege pangozi utano uye sarudza yakasiyana tsandanyama relaxant, izvo kuzvigona zvakanaka mabasa.

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