UtanoGadziriro

Inoshanda antispasmodic "Papaverine Hydrochloride"

Kugadzirira "Papaverine hydrochloride" rinoreva miotropnym zvinoreva kuva simba spasmolytic kushanda. Kwemakumi akawanda emakore, rinoshandiswa kuderedza vascular matauriro uye kumeso tsandanyama kutandara uye zvinenge zvose zvomukati. It ane anzi hypotensive chiito. chinodhaka ichi dilates ari arteries, anowedzera vhoriyamu ropa, kunyanya chepfungwa. Izvi mushonga pamatunhu mishonga zvinoshamisa akazoita excitability pamusoro cardiac tsandanyama, uyewo chinowedzera tava kuderera intracardiac conductivity. simba rake pamusoro nechepakati tsinga kunoratidzirwa zvishoma, kunyange ine kunyaradza kushanda dzakakwirira mishonga.

Tisunungurirei kugadzirira "Papaverine hydrochloride" zvakadaro uwandu husingakuvadzi siyana:

- Mahwendefa nevakura 0,04g (10 hrs.);

- Vana mahwendefa 0.01g (10 hrs.);

- 2% jekiseni (10 ampoules);

- rectal suppositories 20 MG (10 hrs.).

Zvairatidza yokushandisa ndizvo zvinhu zvakadai spasm kuti mvere tsandanyama nhengo peritoneum cholecystitis, renal colic; spastic colitis; endarteriite; bronchospasm; pilorospazme; vascular kurwadza kwacho, iri muuropi. Pakurapa angina pectoris rinoreva "Papaverine Hydrochloride" rinoshandiswa nokuda kukabatanidzwa kurapa nevamwe zvinodhaka.

Contraindications pakushandisa zvinodhaka ichi ndiwo:

hypersensitivity, havachanyatsogoni chiropa basa, yemaziso, pauduku (makore anosvika 0.5). Vakwegura vanofanirwa kutora zvinodhaka uku nekuda mukana hyperthermia.

Rinoreva "Papaverine hydrochloride": mirayiridzo kushandiswa

The mushonga rinoitwa kuti 3-4 p. pazuva. The chipimo chemushonga nokuda kuroora vaitarira mahwendefa kunosiyana-siyana pamwe nemakore murwere. Adults kugadza kuroora dose Mahwendefa 40-60mg. Vana 0.5-2 d - 5mg, 3-4 PM - 5-10mg, 5-6 l. -10mg, 7-9 litres. - 10-15mg, 10-14 litres. - 15-20mg.

Jekiseni chinotarisirwa intramuscularly kana subcutaneously. Majekiseni kuita 2-4 p. pazuva nokuda 1-2ml. Intravenous mushonga jekiseni zvishoma nezvishoma panguva 20mg kare achiwedzera kwachiri yavaibvisa chloride 10-20ml (0,9% mhinduro). nzira iyi zvakanakisisa kuitwa pasi pokudzora chiremba. Varwere vakwegura chete kwokutanga dose haafaniri kupfuudza 10 MG. Kazhinji mushonga chinotarisirwa parenterally akabatana siyana zvinodhaka spazmaliticheskimi uye marwadzo, akadai mushonga "Promedol".

Makenduru vane papaverine raitongwa rectally, 2-3 p. 20-40mg pazuva.

Kugadzirira "Papaverine hydrochloride" anogona kukonzera marwadzo akadai hope, neutachiona, ventricular arrythmia, upregulation kuti chiropa transaminases, BP, kupatira, eosinophilia.

Kana ovhadhozi aona zviratidzo zvakadai vakawanda simba, diplopia, hypersomnia.

Nokushandisa mirayiridzo inokosha iyi kuchengeta mushonga kuti vanokurudzira kungwaririra kushandiswa zvinodhaka vasingadzoreki kuvarwere uye vakwegura; vanhu vane kukuvara mumusoro, hypothyroidism, adrenal dysfunctions, itsvo uye chiropa; tachycardia; kugwinha ezvinhu.

Drug "Papaverine hydrochloride" panguva yepamuviri uye panguva kudyisa nani kwete kushandisa nokuti ayo efficacy uye yakachengeteka yakadaro nguva haina kugadzwa.

Panguva kurapa, doro hakubvumidzwi. Kusvuta panguva kurapwa yekudyidzana akazoita kubudirira chezvinodhaka. Pamwechete kubvuma kunoreva "Papaverine" uye "Dopegitom" chiito chokutanga yekudyidzana ipfupi.

Papaverine hydrochloride Rinowanikwawo vanoverengeka aibatanidza antispasmodics akabatana nevamwe zvinodhaka zvinhu:

- zvinodhaka "Lyupaverin" - pamwe phenobarbital;

- zvinodhaka "Pafillin" - pamwe platifillin gidrotata;

- gadziriro "Kellatrin" - pamwe kellinu uye atropine sulfate ;

- zvinodhaka "Kelliverin" - pamwe Kellin;

- gadziriro "Nikoverin" - pamwe nicotinic acid.

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