UtanoKugadzirira

"Tsinarin": mirayiridzo yekushandisa, kuongorora, kufanana

Calcium channel blockers inonzi boka rakasiyana-siyana remishonga ine mhando imwechete yekuita, asi yakasiyana mune zvimwe zvinhu, kusanganisira kinetic parameters, kusarudzwa kweiviri uye zvinoitika pamutambo wemwoyo.

Nheyo huru yekuita kwemishonga yakadai ndeyokuti vanogona kudzivisa kupindira kweC Ca ions kubva munzvimbo yepislular kusvika mutezi weropa nemwoyo yemasero masero kuburikidza nemakiramuumamato (slowly). Izvi zvinotungamirira kune chirevo chakataurwa chevasodilating.

Uyu anonyanya kuzivikanwa nenyasha ye calcium ndiyo mishonga "Tsinarin." Mirayiridzo yekushandiswa, mari, kuongororwa uye kuumbwa kwechigadzirwa ichi zvicharondedzerwa pasi apa.

Chimiro chekusunungurwa, kuiswa mukati, tsanangudzo, kuumbwa

Mushonga we "Tsinarin", unongororongedzera pamusoro pezvakanaka, unoenderera mberi uchitengeswa nenzira ye biconcave, yakazara uye mahwendefa machena. Chavo chikuru chikamu chinonzi cinnarizine. Mukuwedzera, mushonga unosanganisira zvinokonzerwa nemuviri we povidone K25, lactose, gorosi starch, silicon dioxide colloid uye magnesium stearate.

Iwe unogona kutenga ichi chigadzirwa mumasero emakona.

Mamiriro ekugadzirira

Mirayiridzo yekushandiswa kwechirwere "Tsinarin" inoshuma kuti iyo inopikisana nemasikiramu emagetsi (anonoka). Iyo inoderedza kudengenyeka kwe Ca ions mumasero uye inoderedza nhamba yavo muchitoro che plasmolemma, uye inowedzerawo vasodilating effect ye carbon dioxide uye inoderedza inzwi remuviri weArterioles.

Nokukanganisa zvakananga nemidziyo, ichi chinodhaka chinoderedza kupindura kwavo kune zvinovaka muviri (norepinephrine, adrenaline, angiotensin, dopamine uye vasopressin). Inofanirawo kucherechedza kuti mishonga iri mubvunzo ine vasodilating properties, kusanganisira maererano nemidziyo yeuropi. Muchiitiko ichi, hazvina kuchinja BP.

Mushonga we "Tsinarin", mutengo waro unoratidzwa pasi apa, unoratidza kuenzanirana antihistamine basa, kunoderedza kusagadzikana kwezvigadzirwa zvevastibular uye kunoderedza inzwi rekunzwira tsitsi NC. Ichi chiremba zvinonyatsozviratidza mukukanganisa kwokutanga kwepfungwa yepamusoro, uye mukusingaperi. Mune vanhu vane simba rakaoma rekupararira, inovandudza ropa rekutengesa kwezvinhu zvose uye nhengo. Iyo inowedzerawo kutapukisa kweropa, inowedzera kuwedzera kweyerythrocyte membrane uye musimba kumirisana ne hypoxia.

Kinetics wezvinodhaka

Ndezvipi zvinyorwa zvinowanikwa zvechirwere "Tsinarin"? Mirayiridzo yekushandisa inotaura kuti mishonga iyi yakagadziriswa mumatumbo uye mudumbu. Nhamba yepamusoro yekutungidzirwa kwayo mu plasma inosvika mushure memaawa matatu. Kubatana kwe cinnarizine ne plasma mapuroteni ndeye 91%. Chirwere chacho chakanyatsoshandiswa muropa. Hupenyu hwayo hupenyu maawa mana. Pane mishonga ine urini nemhuru.

Zviratidzo

Mushonga we "Tsinarin" unoratidzwa kutorwa pa:

  • Senile dementia;
  • Ischemic stroke;
  • Craniocerebral trauma;
  • Post-stroke inotaura (kusanganisira chirwere chakanyanya);
  • Discirculatory encephalopathy;
  • Nokudzivirira kinetosis (gungwa kana kurwara kwemhepo, uye panguva yekurwara kwekufamba);
  • Matambudziko eVestibular (kusanganisira chirwere chaMeniere, ruzha munzeve, chizuru, nystagmus, kurutsa uye kushungurudzwa kwe labyrinthine kubva);
  • Migraine (nekuda kwekudzivirira kukanganisa);
  • Kurwisana kwemhirizhonga kupararira.

Kupindirana kwekutora mahwendefa

Ndezvipi zvisingakwanisi kupa mishonga "Tsinarin"? Mirayiridzo yekushandisa inozivisa kuti mhinduro iyi inopesana kana:

  • Hypersensitivity;
  • Kutakura kwe fetus;
  • Kuberekwa.

Inofanirawo kuonekwa kuti ichi chinodhaka chinotarisirwa nekuchenjerera muPalinson's disease.

Kugadzirira "Tsinarin": mirayiridzo yekushandisa

Tora mapiritsi aya anofanira kuva mukati, kunyanya mushure mekudya.

Kana kupararira kweropa kweropa kuchivhiringidzika, mushonga unorayirirwa muhuwandu hwe25-50 mg katatu pazuva, uye munyaya yekusakatika kwemhepo inopararira - 50-75 mg uye yakawanda yakawanda.

Nekushungurudzika kwemavara, mushonga unorayirwa kutora 25 mg katatu pazuva. Ne kinetosis kana iyo inonzi "marwagwa" chirwere, varwere vakuru vanorayirwa 25 mg yemishonga 30 maminiti musati pomugwagwa. Kana zvichidiwa, mushonga wacho unotorwa zvakare mushure memaawa matanhatu (mumutengo wakafanana).

Kuvana, ichi chinodhaka chinorayirwa muhuwandu we22 dose kubva kune munhu mukuru.

Nekunzwisisa kwepamusoro kumishonga, kurapa kunotanga nehafu yesero, zvishoma nezvishoma kuwedzera. Nzira yekurapa inogona kupera kubva pamasvondo 2-3 kusvikira mwedzi yakawanda.

Zviitiko zvakashata

Ichi chinodhaka chinogona kukonzera kuitika kwemashure anotevera:

  • Dry mouth, indigestion, kurwadziwa kwepamuviri, cholestatic jaundice;
  • Kutsiva, kuora misoro, kuneta uye zvinokonzerwa nekuwedzera (semuenzaniso, kuwedzera kwematomu, kutenderera kwechimiro, hypokinesia);
  • Tsvuku tsvina yakachena, kutuka, lupus-like syndrome, rash rash;
  • Allergic phenomena, kuwedzera pfuma, kuderedza ropa.

Mutengo, chibereko chinobudiswa, zvakafanana uye kuongorora pamusoro payo

Kusunungurwa kwezvinodhaka zveboka re calcium channel blockers kunoitwa maererano nemirairo yechiremba. Mutengo wemishonga iyi inenge 20-50 rubles.

Kana zvichidiwa, ichi chinodhaka chinogona kuchinjwa nemishonga: Vertizin, Diziron, Stugesin, Stugeron, Cinazine, Cynedil, Cinnarizine, nezvimwe.

Vazhinji vashandisi vanotora muvengi uyu vanoti iyo inoshanda chaizvo uye inoshanda. Kugamuchira "mahwendefa e" Tsinarin "kunobatsira kugadziriswa kwekushungurudzika kwemaziso uye kushungurudzika mukushandiswa kwekuparadzirwa. Mukuwedzera, mushonga uyu unofadza kunokanganisa muviri wemunhu mu migraines, senile dementia uye post-stroke states.

Inofanira kuonekwa zvakare kuti mhinduro iyi inowanzokonzera maitiro akafanana. Kuti vadzivise kukura kwavo, mazano ose echiremba anofanirwa kunyatsoongororwa. Kutora mahwendefa "Tsinarin" mukuchenjera kwahwo kwakarambidzwa. Vanofanira kunyorerwa chete nechiremba anoenda.

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