UtanoGadziriro

Drug 'Atenolol Nycomed'

Nokuti mushonga "Atenolol Nycomed" pane makemikari, uye international nzvanyira nezita "Atenolol". Mumutauro mishonga pharmacologists zvayakaita zvinodhaka hunoratidzika (RS) -4- (2-hydroxy -3- (isopropylamino) phenyl-acetamide. Tablets "Atenolol" dzinomirira oboevypuklye zvemapuranga mapiritsi ose chena ruvara, vane Kamudzira chimiro. The muviri chikuru anopiwa notch nokuti yokumbozorora rumwe rutivi, pane zviratidzo AV55 uye AV57.

Mune imwe piritsi, zvichienderana kusunungurwa fomu ingasanganisira mashanu kana zana milligrams pakati atenolol. Ebetsero zvinoriumba inoshandiswa talc, gelatin, propylene glycol, titanium dioxide, magnesium stearate, ipromeloza 2910 (15sP), chibage starch, yavaibvisa lauryl sulfate, rinorema magnesium carbonate.

Medicine "Atenolol Nycomed" mabasa somunhu beta1-zvokusarudza (cardioselective) adrenoceptor ichivharira mumiriri, Kamudzira pakudzikamisa basa hakusi. chokushandisa ichi zvinoratidza antianginal, antiarrhythmic uye hypotensive kushanda. It anokwanisa ichivharira Beta-adrenergic receptors mwoyo, kuderedza myocardial kweiyi aimunzwira tsitsi nokupesana autonomic tsinga uye catecholamines, izvo tenderera muropa. Medicine "Atenolol" kwakabatsira mukuderedza sinus automaticity, normalizes mwoyo mwero kuti standstill uye panguva yechiitwa. Izvi nechokumusoro muitiro uye excitation pamusoro myocardial contractility, tava kuderera kubatsira AV-conduction. In kushandisirwa pane kuderera myocardial okisijeni kudiwa. Zvakanaka kunokanganisa hurongwa kushandiswa mishonga "Atenolol" riri BP. Kudzikamiswa of antihypertensive kushanda kunoitika pakazopera vhiki kugamuchirwa wechipiri.

Kugadzirira "Atenolol Nycomed" pamusoro nomumukanwa kugamuchirwa nzira anokwanisa kunakidzwa zvomudumbu turakiti bhuku 50-60% of raitongwa dose. Yabudiswa muna weti pamwe nehafu-upenyu maawa 6-7. Idzi nguva vari varwere renal vanotaura, zvichienderana mwero glomerular filtration.

Zvairatidza kuti zvinodhaka ndiko "Atenolol Nycomed" ndiwo marudzi neBP uye tachyarrhythmias (kusanganisira sinus). Shandisa mishonga uye kuzvidzivirira mumiririri kuti angina kurwiswa.

The daily chipimo chemushonga zvinodhaka nevakura pakurapa angina uye BP rinosvika 50-100 MG. Mahwendefa kubvuma rinoumbwa kusvika kaviri pazuva tichifunga nezvokuti zuva nezuva dose haafaniri kupfuudza 200 MG. Kusuka pasi mushonga inofanira kuva zviduku yakawanda mvura.

The mushonga rinoshandiswa zvichinyatso enderana kunenge ari kupinda chiremba. Dzokuzvirapa haabvumirwi. The mushonga "Atenolol Nycomed" ane marwadzo. Kumwoyo anogona kupindura zvinenge bradycardia, AV-conduction vachivavhiringidza, unogona kuona nezvekufadza ose paresthesia uye Mbabvu inotonhora, mune zvimwe zviitiko pachena zviratidzo mwoyo kukundikana. Zvomudumbu turakiti ikasakendenga nezvinenge zvinodhaka kuda kurutsa, kupatira, manyoka, muromo yakaoma (zvisingawanzoitiki), kuti kwemakemikari anobudiswa hurongwa - pangava kukura munhu hypoglycemic ezvinhu mune varwere vanenge cheshuga, urogenital maitiro - zvinoita kuderera potency. CNS nenjodzi vangapikisa mu musoro, dzungu, hope zvirwere, kuora mwoyo, kunzwa kuneta. Zvinogonekawo neutachiona, kuvaviwa, uye akatsvuka. Nyaya amplification ziya, zvinoderedza kuti misodzi mvura secretion akanyorwa, panowanikwa conjunctivitis.

Uyewo, pane vakawanda contraindications. In dzavo mazita anosanganisira munhu zvokukura chisingaperi mwoyo kukundikana, bradycardia, hypotension, rakawedzera aikanganiswa mushonga, uye vamwe.

Chengeta mishonga panzvimbo yakaoma, kudzivirirwa chiedza, achisiya vana. Room tembiricha 25 ° C. A mushonga anoramba ehupfumi ayo kwemakore mashanu.

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