UtanoGadziriro

"Katadolon": mirayiridzo kushandiswa, mutengo, uye wongororo. Analog "Katadolona"

Chii chinodhaka "Katadolon"? Analogs, mutengo uye mirayiridzo kushandiswa kwezvinodhaka zvichakurukurwa munyaya zvinhu ino. Mariri uchadzidza, uye kuti chii chinorehwa inzira, kana vane chero contraindications uye marwadzo, mune ipi aripo kuti rine wayo marongerwo uye zvichingodaro.

Kavha, kusunungurwa siyana, akafanana

Drug "Katadolon" anoenderera mberi Sale zviviri zvakasiyana siyana. tsananguro dzavo, akafanana uye kavha, tinotarisa zvino.

  • Medicament "Katadolon Forte" - yellow biconvex denderedzwa mahwendefa (rimwe divi ubvise) ine zvakasiyana siyana inclusions. Kugadzirira rine kutoshanda pakuderedza sezvo flupirtine maleate, uye dzimwe Excipients. Mahwendefa anoiswa mukati Maronda akasiyana 10, 7 uye 14 zvidimbu, izvo mumapepa ari packs it kuti makadhibhokisi.
  • Capsules "Katadolon kutadzisa" sheathed mu tsvuku gelatin. The zviri zvinodhaka ari guruva rinopfumburwa yero-nyoro kana tsvuku Hue. Mumwe Kamudzira rine flupirtine maleate, uye mamwe vamiririri sezvo gelatin, magnesium stearate, mvura, titanium yakasviba E172, nesilicon dioxide, yavaibvisa lauryl sulfate, dihydrate karusiyamu phosphate uye copovidone. The mushonga ari mumapepa mu packs it pamusoro makadhibhokisi 30, 50 kana 10 capsules.

The pharmacological zviito zvinodhaka

Chii sechinhu zvinodhaka uye kana ane analoginen? "Katadolon" - asiri opioid unonyaradza marwadzo kuti ane antispasmodic chiito, uye aine muzvizhinji kuti analogues siyana.

Mishonga haisi muropa uye anokwanisa kupa centralized zvazvinoita. Mushure kudya kwayo kunokanganisa G-mapuroteni, nokudaro vachichinja zvinogona musiyano iri karusiyamu hova uye pakudzikamisa nyika neuronal Kamudzira zvinogona.

Zvakaita nzvimbo yacho vaiona medicament yayo ishamwari? "Katadolon" zvinofanira kutorwa mu mishonga kuti haapfuuri kufadza zvinobvumidzwa. Chete muchiitiko ichi chacho vanoshingaira chirungiso asingadi kukanganisa H uye M-cholinergic receptors, uyewo opioid, dopamine, kweserotonin, uye alfa2- alpha1-adrenergic receptors.

Pamusoro pokugamuchira capsules kana mapiritsi mukati analgesia kunoitika anoonga Kuziviswa potassium migero, izvo zvinowanikwa mumasero tsinga.

Maererano nenyanzvi, mishonga yakanaka nomugumisiro NMDA-receptors. Iye anomira matsva calcium ions, izvo nomunyika semipermeable Kamudzira rusvingo.

Pfungwa chiito ane mushonga

Sei muviri womunhu inotaura nzira yayo ishamwari? "Katadolon" rine aro Zvinoumba flupirtine. Hazvina fuma iyi kunodzivisa etsinga chido ikarumbidzwa kune nociceptive kuitika. Somugumisiro dzokuteerera kwakadaro kunoitika yokutindivadza.

The mushonga hariwaniki zvinorwadza nezvekufadza uye kunotadzisa kubva kuva refu. Uyezve, zvinobudirira nayo lowers vane marwadzo.

Pamusoro anogamuchira zvinoreva kupinda tsandanyama kutandara kunoitika (nokuda ichivharira pamusoro zvenguva Tutsinga tunofambisa mashoko utwu). Hatigoni kutaura kuti zvinodhaka izvi anokwanisa kudzivirira Tutsinga tunofambisa mashoko utwu kubva zvinokonzerwa muchetura. Simba karusiyamu Mipata medicament akazoita zviri anokuvadza karusiyamu ions ari mumasero.

The pharmacokinetics zvinodhaka

At okutambirwa mahwendefa uye capsules "Katadolon kutadzisa" iri gastrointestinal zvinodhaka vanoshingaira fuma wefodya zvachose (anenge 90%). Saka 75% of dose rinoita mune chiropa.

The hafu-upenyu muviri ndiwo maawa 7-15. 70% of zvinodhaka yabudiswa parutivi netsvo, uye vamwe - kuburikidza muura.

In vakwegura, uye varwere havachanyatsogoni chiropa nerevane itsvo kubviswa hafu-upenyu inowedzerwa.

Drug "Katadolon": zvairatidza yokushandisa

The zvairatidza kuti kushandisa zvinodhaka ichi vari kurwadziwa siyana mavambo (nepakati), izvo zvinokonzerwa spasm kuti mvere tsandanyama.

Saka pasi chero zvarakasiya ushandiswe vaiona nzira yayo ishamwari? "Katadolon" rinowanzoshandiswa post-kushanda marwadzo uye kutemwa nomusoro, kurwadziwa uye mutsipa, nyanyisa neoplasms uye namamota, uye zvichingodaro. D.

Contraindications pakushandisa zvinodhaka

Medicine "Katadolon" haisi varumbidzwa kushandisa kuti itsvo uye chiropa, hypoalbuminemia, nezvimwe zvinhu kuti basa chirungiso kana ebetsero zvinhu, tinnitus, uyewo pakurapa vakwegura, vana uye zvidhakwa.

Dosing medicament

Ndinofanira kutora mishonga "Katadolon"? Capsules chero zvazvingava hazvibviri kutsenga. The chipimo chemushonga zvinodhaka anosarudzwa chete nomunhu.

Zvinotevera regimens anopiwa mune dzakabatanidzwa mirayiridzo iri medicament:

  • Vakuru kusvika makore 65 ushandiswe 100 MG zvinodhaka kanokwana pazuva (kureva 1 Kamudzira). Zvinofanira kuomerera iyoyo zvikamu pakati zvinodhaka mishonga. Kana akaratidza marwadzo chirwere anobvumirwa kutora capsules maviri katatu pazuva. Zvinofanira kurangarirwa kuti kufadza zuva chipimo chemushonga inofanira kuva MG 600 (i.e. 6 capsules).
  • Vakwegura (anopfuura 65 years) zvinodhaka "Katadolon" vanofanira kutora 100 MG kaviri pazuva. Zvichienderana mwero marwadzo dose anogona ngazviwedzerwe 300 MG pazuva.
  • Varwere vanotambura renal insufficiency kana hypoalbuminemia, kazhinji dzakabatwa asingapfuuri 300 MG pazuva.
  • Kana medicament vasingadzoreki chiropa basa haigoni kubatwa mishonga, iyo kupfuura MG 200 pazuva. Ya kurapwa ichi angava akasiyana. Zvisinei, pamwe kwenguva refu kurapwa kunodiwa kudzora basa chiropa makemikari.

Analogs "Katadolon" chinodhaka ane chete rinoita wemafuta sezvo chepakutanga. Zvisinei, kana vari dzakasarudzwa se yokutsiva, iva nechokwadi kuti bvunza chiremba wako uye kusarudza optimum chipimo chemushonga.

Ovhadhozi zvinodhaka

Kune Mishumo shoma nyaya zvinodhaka ovhadhozi "Katadolon" nevavariro kuzviuraya. Muchiitiko chino, waunowana zvinotevera zviratidzo: svoto, mumamiriro prostration, tachycardia, kuvhiringidzika, vachidanidzira, kuoma muromo, vakashamiswa.

Mukurapa zviratidzo zvakadai kushandiswa diuresis. Uyezve, mumwe murwere inopiwa kusashanda kabhoni uye electrolyte nezvevanakomana. Subject nezviyero zvose izvi murwere nemamiriro anovandudza pashure pemaawa 6-12.

Nenjodzi pashure ingestion

Vamwe varwere pashure ingestion mahwendefa kana "Katadolon" capsules ngaakuitireiwo zvakadai nemishonga se:

  • dzungu, simba, uye nekuneta;
  • flatulence, kuda kurutsa, uye abdominal kurwadziwa;
  • tremor, fufune;
  • nomusoro uye kunetseka;
  • neutachiona;
  • zvinodhaka Kutemeswa chiropa;
  • madzerere.

Nemishonga zvingaitika risingatarisirwi uye pakarepo kunyangarika uyewo paaiita mishonga.

zvinodhaka kwavatori

Apo mawa Kutarisirwa "Katadolon" kugadzirira zvinoreva akadai "Warfarin" uye "Diazepam" wokutanga chiito anogona huchawedzerwa. Izvi imhaka yokuti zvinodhaka izvi vasunge nyore chete mapuroteni inotsigira misha masero flupirtine.

Sedatives, tsandanyama relaxants, uye panyaya iyi kusimbisa migumisiro zvavo pasi pokudzora mushonga.

Hazvina varumbidzwa chokubatanidza mushonga ne "paracetamol", "carbamazepine" uye "flupirtine."

Zvinofanira kucherechedzwa kuti apo kushandiswa zvinodhaka "coumarin" zvakafanira kuongorora prothrombin indekisi.

Zvokungwarira

Asati kushandisa mishonga, "Katadolon" vanofanira kuverenga rairo. Rinotaura kuti:

  • mushonga uyu anofanira kushandiswa chete kana zvimwe inonyaradza marwadzo omusoro ARV contraindicated.
  • Panguva pokushandisa medicament mune vanhu vane akaderedza itsvo basa zvinokosha kudzora wevasungwa pakati creatinine muropa.
  • Persons vakuru makore 65 uye varwere hypoalbuminaemia uye zvakakomba renal vanotaura vanoda dose kuchinja zvinodhaka.
  • Varwere vanofanira kunyeverwa kuti panguva mushonga vanofanira kubhadhara pfungwa zviratidzo chiropa chirwere. Kana kuratidza zviratidzo zvakadaro vanofanira kurega kutora zvinodhaka uye chiremba.
  • Panguva mushonga mushonga "Katadolon" zvichibvira zvenhema zvakanaka bvunzo paakasangana urobilinogen, bilirubin, uye mapuroteni iri weti.
  • Kana kushandisa yakakwirira mishonga zvinodhaka ari murwere anogona kuonekwa weti staining rwegirini. Izvi hazvisi chiremba chiratidzo ane chirwere.
  • Panguva kurapwa zvakafanira kusiya michina uye motokari kutyaira masimba, sezvo varwere zvingamuka dzungu uye hope.

Drug "Katadolon": analogues, wongororo, mutengo

It kwakafanana ne sando pakugadzirira "Flugesik". Kana akasiyana, yevaifungidzirwa zvinosanganisira zvinotevera mishonga: "Acupan", "Nefopam", "Milistan" uye "Sinmeton".

Price vaiona mushonga chaizvo. Kazhinji, yemakomo 900-1200 rubles (zvichienderana chimiro uye nhamba mahwendefa, capsules).

Maererano mhinduro wevarwere, mishonga "Katadolon" zvikuru zvinobudirira uye nokukurumidza chero vapi marwadzo syndromes. Pasinei vakawanda nenjodzi, vakapindwa muropa nezvinodhaka vanowanzoshandisa ichi sechekushandisa kurwadziwa panguva kurega.

Kana varwere vanhuwo, vamwe vavo vanotsutsumwa kuti kutora zvinodhaka uku kunowanzoita dzungu uye zvayo neutera.

Maererano vanachiremba, mushonga "Katadolon" rinowanzoshandiswa kuvhiya tsika. Iye simba zvikuru, saka hazvifaniri kutorwa pasina chiremba mushonga.

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