UtanoGadziriro

Makenduru "Proktoglivenol": nhoroondo, mirayiridzo kushandiswa, analogs

Ko "Proktoglivenol" makenduru kubatsira? Reviews ari kubudirira zvinodhaka izvi zvichakurukurwa pazasi. Uchadzidzawo sei mushonga uyu unoshanda, umo nguva zvinonzi ushandiswe, zvakadini tinorasikirwa uye kana analogs.

Kavha, akafanana

Makenduru "Proktoglivenol" mirayiridzo kushandiswa iro raiva panzvimbo makadhibhokisi pasuru, akapisira kutengeswa muna mhoni packs it 5 zvidimbu. Yatochena oblong suppositories kuti rectal kutarisira uye anosanganisira ayo nhengo dzakadai unorapa sezvo tribenozid uye lidocaine. Uyewo gadziriro ino ine ebetsero zvinoriumba Witepsol E85 uye Witepsol W35.

Hatigoni kutaura kuti kutengeswa angawana imwe chimiro zvinodhaka. "Proktoglivenol" - okuzora chena, homogeneous, opaque uye kuva yakananga kunhuwa. Inowanika ane 30 d chubhu uye rine zvakafanana vanoshingaira zvinoriumba.

Key ehupfumi

The mushonga "Proktoglivenol", mitengo yakanga dzichakurukurwa pazasi, rinotarisirwa kuti kukamura uchishandisa mishonga Mamota. Rine unorapa maviri - lidocaine uye tribenozid. Nemhaka zvavo pamberi, mishonga anokwanisa kupa venotoniziruyuschee, dzomunharaunda rufimbi uye Anti-anogumbura mugumisiro. Rinotaurawo anovandudza microcirculation, kunoderedza marwadzo uye kusimba kuzvimba.

Parinoshandiswa pana varumbidzwa dosages makenduru akacherekedza kuderera venous kuzara, kuderera vascular permeability uye kubviswa zvisingafadzi zviratidzo zvakadai Mamota kuvaviwa uye kurwadziwa mugaranhoko uye horo.

musimboti oparesheni

Kuchirapa nemigumisiro uye mashandiro kuita zvinodhaka pasi kukurukurwa zvinokonzerwa pharmacological zvechadenga vanoshingaira zvinhu zvayo sezvamunoita.

Sezvo pane "Proktoglivenol" makenduru? Mirayiridzo dzokushandisa inoti tribenozid chinhu chakaita zvokugadzirwa fuma kungova kirasi glyukofuranozidov. mashandiro ayo chiito haina aizvinzwisisa. Zvisinei, nyanzvi dzinoti kuti inobatanidzwa vachikwanisa tribenozida mwoyo simba basa endogenous amines akadai histamine, bradykinin, uye kweserotonin.

Hatigoni kutaura kuti inzira antagonist tribenozid humoral zvinoita kuti pave nokuda edema, vasodilatation, vakawedzera permeability midziyo ropa uye kuzvimba.

Munguva yokudzidza zvakanzi akacherechedza kuti zvinodhaka "Proktoglivenol" (mafuta uye suppositories) hakurevi kukanganisa basa endogenous vasoconstrictors kusanganisira norepinephrine uye epinephrine. gadziriro iyi anobvisa kuzara ari mutsinga, asi kunowedzerawo matauriro avo uye anoderedza yakakwirira (pathologically) vascular permeability.

Kusuma ane antagonist kuti anogumbura nevamiririri tribenozid application kunoderedza kusimba kushoma, ane Anti edema uye marwadzo anokonzerwa. Zvinofanira kucherechedzwa kuti fuma iri mubvunzo kunoderedza mano maplatelet kuomerera.

Chii muchinangwa zvinodhaka lidocaine "Proktoglivenol" (mutengo chokushandisa ichi kuwanikwa vose)? chaikosha uyu munharaunda rufimbi mumiririri, iyo inesungano nomukaka zviri acetanilide.

The kushanda nhungamiro vakati rinoreva hwakavakirwa kukwanisa kwayo chaivharidzira yavaibvisa migero, zvichiguma pakudzikamisa muchitokisi membranes.

Nyanzvi dzinoshuma kuti lidocaine kuchititadzisa chizvarwa zvakanaka, uyewo conduction kuti nomunhu ari etsinga fibers. Muchiitiko chino, pane zvikuru sei maitiro ake uye marwadzo nomunhu, nomunhu nezvimwe modalities.

Mukuita zviri muvanhu mubvunzo kukamura uchishandisa kushanda asina zvainoita myocardium.

Kinetic zvechadenga gadziriro

Ko "Proktoglivenol" makenduru vari kunyura? Reviews vanoti mushonga uyu kana raitongwa rectally tribenozida bioavailability anenge 30% kuti kana uchishandisa dzinogamuchidzanwa Formulations pamwe chete rinoita fuma.

Peak yeplasma kuwanda tribenozida kana rectal Kutarisirwa anenge 1 ug / Rine mamiririta. ukoshi iyi yakasvika pashure 2 maawa pashure kwokubatsira suppositories.

Kana dzemauto "Proktoglivenol", kana rinoshandiswa munyika anopinda muropa pamusoro 5-20% tribenozida. Tribenozida muviri kunoitika muna chiropa uye yabudiswa ainyanya sezvo metabolites neitsvo.

Maererano mirayiridzo, lidocaine nokururamisira zvakanaka kunyura kana kushandisa dzemauto pamusoro mucous membranes. Zvinofanira kucherechedzwa kuti pashure kubvunza sanganisika ganda Absorção de Água izvi zvinhu yakaderera.

Pashure rectal suppository lidocaine bioavailability anenge 50% uye yepamusoro yeplasma wevasungwa - anenge 0,7 ug / Rine mamiririta (kubudirira mumaawa maviri).

umboo

"Proktoglivenol" Ko sei makenduru? Reviews akashuma kuti chokushandisa ichi ari kushingaira kushandiswa nokurapwa yomunyika uye zvimwewo Mamota vanhu vane mwero zvakakomba uye zvine mwero weboka chirwere.

Zvinonzi zvakare nezvenzvimbo mushonga inogona kushandiswa pakurapa varwere zvikuru Mamota kana chipi chikonzero hapana mukana wokuita kuvhiyiwa.

Contraindications

Ita contra "Proktoglivenol" makenduru? Nyanzvi Guest vanoti kuti dzairambidzwa basa redu kushandiswa kwezvinodhaka ichi zvishoma. Akanga asina vakagadzwa chete zvinotevera nyaya:

  • ari trimester akazvitakura rokutanga;
  • dzakakwirira aikanganiswa pezvokuvamba zvinodhaka;
  • vana (nokuda kwokushayiwa yakavimbika mashoko pamusoro zvinodhaka kuchengeteka uye efficacy).

Ndingatarira kushandisa makenduru kubva Mamota "Proktoglivenol"?

Reviews wevarwere yakataura kuti mishonga hunoratidza inoshanda chete kana mukanyatsochengeta kutevedza mazano ose chiremba.

Viewed mushonga unoshandiswa rectally. zviri pamberi chakaunzwa ari mumagaro Canal inofanira kuva zvakasimba maoko enyu.

Duration yokurapa uye chipimo chemushonga zvinodhaka chete kunotema chiremba nomunhu.

Kazhinji, vanhu vakuru kukura chakasimba Mamota zvinodhaka kugadza 1 suppository kaviri daily (kana 1 kushanda mafuta). Kurapwa vakatakudzwa kubva mangwanani uye manheru, kusvikira wakakwana kunyangarika iri rikwanise zviratidzo.

Kana chiremba mufananidzo inovandudzika, uye kupera vose salient zviri maperembudzi, yezwi kushandisa makenduru 1 kana 1 kushandiswa mafuta kamwe pazuva.

varwere Adult pamwe kukura yomunyika Mamota vaiona zvinodhaka iri chinotarisirwa ari muchimiro ruomba kana suppositories kuti mureza muenzaniso. Panyaya iyi, namafuta inokurudzirwa chinofanira kutarisirwa zvakananga kupinda mugaranhoko uchishandisa chaiyo applicator.

Zviito zvakaipa hunhu

Kugadzirira Mamota "Proktoglivenol" zvakanaka akashivirira nevarwere. Dzimwe nguva pamusoro kushandiswa kwayo muvanhu vakachengeta romunzvimbo neutachiona, kusanganisira ganda kuvaviwa. Uyewo, zviri zvisingawanzoitiki zviitiko, kushandiswa mishonga, varwere chema unopfuta manzwiro ari horo.

Drug "Proktoglivenol" (makenduru) paanenge achiyamwa uye panguva pamuviri

Maererano mirayiridzo, kuti medicament mu mubvunzo inogona kushandiswa panguva lactation. Zvisinei, izvi zvinofanira kuitwa chete mushonga ari kupinda chiremba.

Ndinogona kushandisa zvinodhaka "Proktoglivenol" (makenduru) panguva pamuviri? chokushandisa ichi haina yakarumbidza panguva mitatu yokutanga gestation. Mune trimester wechipiri nowechitatu, unogona kurongera izvozvo, asi chete kana zvinobatsira kuti mai kudarika yavanababa zvingakanganisa mwana.

zviitiko ovhadhozi

To musi, hapana mishumo ovhadhozi pakati mari kunge kugamuchirwa.

Kana mushonga yakanga netsaona anwa kubudikidza murwere, ipapo vanoita kwokukurumidzira gastric lavage, uyewo vakanzi kugamuchira enterosorbents. Kana waida kuti rinoitwa uye symptomatic kurapa.

Mari chinodhaka, analogues ayo

Chii mutengo uye chii unogona kutsiva mishonga «Proktoglivenol" (makenduru)? Analogues, mutengo zvinodhaka izvi zvichakurukurwa zvino.

Kana mumwe chikonzero kana mumwe mari haazopindi, panzvimbo pake zvinodhaka zvinotevera zvinogona kushandiswa Mamota "Anuzol", "Bezornil", "Relief Pro", "Betiol", "Proktozan Neo", "Pileks", "Proctosedyl "" Proktan "," Relief "," Gemorron "," Aurobin "Belladonna mushoma," Proktozan ".

Kana mutengo, ipapo kenduru uye ruomba "Proktoglivenol" rinogona siyana. Kazhinji, suppositories vari rubles anenge 400, uye mafuta vanenge 550 rubles.

Reviews zvinodhaka (rectal suppositories nezvizoro)

Reviews ose rectal suppositories vainyanya akanaka. Varwere vanenge hemorrhoid kuzvimba, nharo kuti mashomanana pamazuva mushonga anokwanisa kubvisa zvose zvinoitika nezvekufadza yakafunuka, unopfuta uye marwadzo chokuita nechirwere ichi. Uyewo mushonga zvikuru zvakanaka mumagaro Kunetsana uye akapotsa haambokonzeri neutachiona.

Hatigoni kutaura kuti vakawanda varwere vanosarudza kushandisa mafuta "Proktoglivenol". sarudzo dzavo, ivo kutsanangura chokwadi chokuti rectal suppositories vanoguma zvikuru nokukurumidza uye mafuta inogona kushandiswa kwenguva refu. Zvisinei, iye nokukurumidza uye vakachengetwa inobvisa zvose zvinoitika zviratidzo pamberi pematanho kuzvimba Mamota kwazvo Inowedzera muitiro chokuporesa.

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