UtanoGadziriro

Medicament 'Neostigmine'. Mirayiridzo yokushandisa

Kugadzirira "Neostigmine" (Mahwendefa, majekiseni) chokuita FIs pamusoro cholinesterase. The rinoita zvinoriumba zvinodhaka - methyl sulfate neostigmine.

Chezvinodhaka chinobata kunyanya peripheral ino, yakaoma kupinda neropa-uropi nokuidzivirira. Zvinoratidza mushonga "Neostigmine" mirayiridzo kushandiswa zvinoreva kukwanisa kwayo kuderedza intraocular kumanikidzwa, kuderedza pamusoro vadzidzi. Means chinokurwadzai nokuwedzera matauriro uye contractility pakati anotsvedzerera tsandanyama ari zvomudumbu ino, Árbol uye Urinary dundira, chinokonzera bradycardia, spasm akkommodasie. The mushonga runogonesa ziya, mate uye dzimwe kufanana kwemakemikari anobudiswa mumasero ezvinhu, kunoita kufambisa pamusoro neuromuscular hutachiwana, zvisinei yakakwirira siyana kungaita chinovhiringidza kwayo.

The kuchirapa chipimo chemushonga zvinodhaka "Neostigmine" haina nechepakati simba. Zvakaitwa zvinodhaka kwakacherechedzwa pashure maviri kusvika makumi maminitsi ndichienda maviri nehafu - maawa mana. Zvinoreva kunonyanyisa wevasungwa yakasvika muna mumwe maviri maawa.

Drug "Neostigmine". kunyoresa

Akaratidzawo medicament kana injini zvinetso nokuda kukuvara uropi, encephalitis, poliomyelitis, yomumuzongoza, rutivi rwomuviri. Basa zvinoreva uyewo panguva myasthenic dambudziko, myasthenia gravis, atony (dundira, ura, dumbu). By neuchapupu zvinodhaka "Neostigmine" mirayiridzo kushandiswa uye anotakura ane atrophy pamusoro optic etsinga, neuritis, yemaziso. The mushonga rinoshandiswa sezvo mushonga tsandanyama relaxants.

Dropwise kutarisirwa zuva nezuva 0.5 MG kamwe kana kaviri kuna vakuru, vana - hupenyu 0,05 MG gore (asi kwete kupfuura 0.75 ml ane 0,05% mhinduro).

Inside nayo akataura kutora pazuva 0.015 d maviri katatu. Duration kurapwa - maviri namashanu - mazuva matatu. Kana zvakakodzera, kuzodzosera kurapwa penguva pakati kurapwa makosi - nhatu mana vhiki.

Contraindications kune nzvimbo "Neostigmine" mirayiridzo kushandiswa zvinosanganisira zvokuimba mhingaidzo nezvezvimwe zvinetso zvedundira turakiti kana bowel, peritonitis, nomumwe kusashivirira. Not yakatarwa mumiriri nokuda atherosclerosis, angina, asima, hyperkinesis, netsviyo. Regai kutora mishonga pavanenge vakazvitakura uye lactation.

Zvimwe nenjodzi kana uchishandisa idzidziso "Neostigmine" mirayiridzo Chinyorwa inodaro kuda kurutsa, vakawedzera peristalsis uye spastic rutapudzo ari ura, hypersalivation (kunyanya salivation). The akaipa kuratidzwa zvinosanganisirawo arrhythmia, ziso nenyonganiso, kurasikirwa pfungwa, simba, kufenda, dzungu, atrioventricular nechigumbuso, hope. The mushonga "Neostigmine" kukonzerawo Árbol Kusimbaradza uye pharyngeal secretions, hypotension, cardiac kusungwa. Kwakaomarara kuratidzwa zvinosanganisira uye neutachiona, wakawedzera vangadikitira, kuita weti kakawanda, arthralgia, dysarthria, kugwinha, kurwadza kwacho mu skeletal tsandanyama (kusanganisira rurimi musculature), tremor, bronchospasm, chinovhiringidza (kusvika kumisa) zvokufema, wheezing.

Ovhadhozi mushonga "Neostigmine" akaratidza kakawanda weti, manyoka, wakawedzera motility, kuda kurutsa, chinyamunhari chinorwadza, cholinergic dambudziko. Uyezve, pane twitching pamusoro skeletal tsandanyama uye rurimi tsandanyama, kuwedzera tsandanyama simba, hunoreva kufema netsandanyama. Kusimbisa zviratidzo zveefa ovhadhozi wemishonga "Neostigmine" mirayiridzo zvavakabvumirana Kutarisirwa metatsina, atropine nezvimwe M-anticholinergic nevamiririri.

Zvinofanira kucherechedzwa kuti jekiseni zvinodhaka "Neostigmine" haana chete akashandiswa kurapwa kwevanhu, asi mhuka. In wemhuka, mushonga wacho nachiremba kusagadzikana motokari mabasa.

Asati kushandisa zvinodhaka "Neostigmine" zvinokosha chiremba uye dzinotibatsira pfupiso.

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