UtanoKugadzirira

Zvinoreva "Etaperazin". Mirairo yekushandiswa

Mushonga we "Etaperazin", uyo mutengo wake 250 rubles, inonzi neuroleptic (antipsychotic), piperazine derivative ye phenothiazine. Zvichida, migumisiro yemishonga iyi inokonzerwa nekuvhara mumakumbo ekutorera maziso e-dopamine postsynaptic receptors. Iyo mishonga ine simba rakasimba antiemetic - iyo inyanzvi inoratidzika mukudzivirira kana kudzivirirwa kweD2-dopamine receptors neipi inokonzerwa homoreceptor cerebellar zone, uye mhirizhonga inogadziriswa mumatumbo emuviri we vagus nerve. Mushonga wacho wakasiyana uye alpha-adrenoblocking effect. Sedation uye anticholinergic zvinogona kunge zvisingakwanisi kana kuenzanisa zvakasimba, hypotensive basa haritauri zvakajeka. Mushonga "Etaperazin" (kuongororwa kweyanyanzvi kusimbisa izvi) kunewo unofadza kuitika pamisungo. Antiemetic inoitika inogona kukurudzirwa nemaitiro uye anticholinergics. Kurapa zvinodhaka kunowanikwa kunyanya nemuyo.

Kusarudzwa

"Etaperazine" inokurudzirwa pakurapa kwepfungwa dzepfungwa, pamwe chete nekunakidzwa uye kusagadzikana. Zviratidzo zvinosanganisira schizophrenia, neuroses yakaoma nekutambudzika, kutya. Chirwere ichi chinoratidzwa neganda rekuchenesa, kubvisa kurutsa kana kushungurudzika kwechimwe chiitiko chezviitiko.

Mushonga "Etaperazin".
Mirairo yekushandiswa

Nhamba yakakurudzirwa yevarwere vane makore gumi nemaviri isine 4-80 mg. Pachikonzero chenguva isingaperi yezvirwere, huwandu hwemishonga hunobvumidzwa (pane zvinokurudzirwa weyanzvi) kuwedzera kusvika 150-400 mg. Nguva yekubvumirwa uye kuwandisa kwayo pazuva kunotsanangurwa chete nachiremba.

Zvikanganiso

"Etaperazin" (mirayiridzo inoshandiswa inoshandiswa inonyevera pamusoro peizvi) inogona kukanganisa zvakaitwa extrapyramidal ye parkinsonian uye dystonic mtundu, melanosis, cholestatic jaundice, maonero asina kunaka, photosensitization. Mhedzisiro isingadikanwi inosanganisira akathisia, kuputika kweganda pamwe chete nedermatitis, kurara, kunetseka nekugunzva. Pachikonzero chekurapa zvichida kuvhiringidzwa kwekugara, yakaoma muromo. Kazhinji kune kupiswa kwehupenzi, agranulocytosis.

Contraindications

Zvinoreva "Etaperazin" kurairirwa kwekushandisa hakubvumiri kutungamirirwa muhepatitis, cirrhosis, hematopoiesis, nephritis, hemolytic jaundice, panguva yekubata. Contraindications inosanganisira pathology yemutsipa wepelinha uye uropi hwomutambo we systemic mumutambo unofambira mberi, pamuviri, chirwere chebonchoectatic munguva yekupedzisira, hypersensitivity. Iyo mishonga haina kukurudzirwa kune zvirwere zvepromboembolic, kusagadzikana kwemoyo kwekubhadharwa rudzi. Kuchenjerera pakurondedzera mishonga "Etaperazin" (mirayiridzo yekushandiswa ine data yakadaro) kuratidzira nehosha yaPasinson, kudhakwa doro, kushungurudzika kwechiropa basa. Kugadziriswa kwezai kunogona kudiwa kana pane chikonzero chekuitika kwe glaucoma, kuora mwoyo kwekurwadziwa, kupora kwechirwere chinopfutidza kupora. Ngwarira kushandisa iyi mishonga mukurapa kwevasina simba, vakapera simba, varwere vakwegura nevana.

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